International Journal of Drug Discovery

Editor-in-Chief :
Publisher : Bioinfo Publications
ISSN : 0975-4423 (Print)     E-ISSN : 0975-914X (Online)     Frequency : Yearly
Index Copernicus Value (ICV) : 7.00 (2012); 4.18 (2011); 4.48 (2010)       CODEN : IJDD
DOI : 10.9735/0975-4423       Abbreviation : Int J Drug Discov
Subject : Pharma

Most Downloaded Articles

Oncoproteomics: New trends in analytical techniques
Girish Gupta, Nikhil Gupta, Mayank Gupta, Soham Trivedi, Prasad Patil, Vamsi Krishna K, Hipal Gaudani, Gomase V.S.,
Volume : 1   Issue : 2,   Year : 2009           Downloads : 1261

A COMPUTATIONAL MODEL OF THE ROLE OF IONIC-LOCK INTERACTIONS IN LIGAND RECOGNITION BY THE HUMAN C3a RECEPTOR
VOLETI S.R.,
Volume : 4   Issue : 1,   Year : 2012           Downloads : 1230

1Synthesis and QSAR analysis of 5-substituted (arylmethylene) pyridin-2-amine derivatives as potential antibacterials
Choudhari P.B., Mulani A.K., Bhatia M.S., Ingale K.B., Bhatia N.M.,
Volume : 1   Issue : 1,   Year : 2009           Downloads : 1229

Study of new developments in birch reduction process and their applications for the synthesis and CNS depressant activity of 3- aminocyclohexa-1,4-diene-1-carboxylic acid and 3-[5-substituted 1,3,4-thiadiazole-2-yl]-2-styryl 5,8-dihydroquinazoline-4 (3H)-ones
Charbe N.B., Mehere A.P., Shende S.G., Mohod V.S., Gautam D.T., Madusudhan M., Chaitanya Ch,
Volume : 2   Issue : 1,   Year : 2010           Downloads : 1218

Formulation and Evaluation of Indomethacin Microspheres using natural and synthetic polymers as Controlled Release Dosage Forms
Chinna Gangadhar B., Shyam Sunder R., Vimal Kumar Varma. M., Sleeva Raju M., Sai Kiran M.,
Volume : 2   Issue : 1,   Year : 2010           Downloads : 1217

Molecular docking and binding energy studies on nuraminidase of h1n1 reveal possible answer to its resistance for oseltamivir
Meshram R.J., Jangle S.N.,
Volume : 1   Issue : 2,   Year : 2009           Downloads : 1205

Comparative modeling of CDP-diacylglycerol-serine O-phosphatidyltransferase in Clostridium botulinum: A potent target of Botulism
Koteswara Reddy G., Mohan Kalyan Reddy K., Nagamalleswara Rao K., Gyana R.Satpathy,
Volume : 2   Issue : 2,   Year : 2010           Downloads : 1166

Drug design based on the principle of conjunction: synthesis, characterization and antihyperglycemic activity study of 3- [2- (3- aroyl- 2, 4- diphenyl- 3 , 4- dihydro- 2h [1, 3] oxazino [5, 6-h] quinolin- 6- yl) ethyl] 2- phenyl- quinazolin- 4(3h)- ones
Singh S., Bishnoi A., Awasthi R., Pandey V.K., Tiwari A.K., Awasthi N.K., Srivastava K.,
Volume : 1   Issue : 2,   Year : 2009           Downloads : 1147

QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIPS (QSAR) OF A SERIES OF KETONE DERIVATIVES AS ANTI-CANDIDA ALBICANS
LUIZ FREDERICO MOTTA, WANDA PEREIRA ALMEIDA,
Volume : 3   Issue : 2,   Year : 2011           Downloads : 1136

CYTOGENETIC TOXICITY EFFECTS OF LOCAL PURSLANE (Portulaca oleracea) LEAF CRUDE EXTRACTS ON NORMAL AND CANCER CELL LINES in Vitro
HAZHA J.H., ZAKARIA A.S.,
Volume : 5   Issue : 1,   Year : 2013           Downloads : 1136

DETERMINATION OF THE EFFICACY OF 600MCG ORAL MISOPROSTOL IN THE PREVENTION OF POSTPARTUM HAEMORRHAGE
PATVEKAR M., GAIKWAD V., CHANDRAWAT S., MULAY P., GARG R., PURI M.,
Volume : 4   Issue : 2,   Year : 2012           Downloads : 1133

L-ASPARAGINASE-AN ANTI TUMOR AGENT PRODUCTION BY FUSARIUM EQUISETI USING SOLID STATE FERMENTATION
KALIWAL B.B., HOSAMANI R.,
Volume : 3   Issue : 2,   Year : 2011           Downloads : 1124

EFFECT OF PENETRATION ENHANCERS ON IN VITRO PERMEATION OF NYSTATIN FROM TOPICAL FORMULATIONS
MARZOUK M.A., AMMAR A.A., DARWISH M.K., EL-SAYED H.A.,
Volume : 4   Issue : 2,   Year : 2012           Downloads : 1099

Antihepatotoxic and antioxidant defense potential of Mimosapudica
Brindha V., Nazeema T.H.,
Volume : 1   Issue : 2,   Year : 2009           Downloads : 1095

Micro-RNA in development
Thikekar V.P., Sawant J.J., More M.K., Nair V.K., Athalekar P., Patil D., Kulkarni S., Gomase V.S.,
Volume : 1   Issue : 2,   Year : 2009           Downloads : 1092

Induction of apoptosis by the aqueous and ethanolic leaf extract of Vitex negundo L. in MCF-7 human breast cancer cells
Arulvasu C., Prabhu D., Manikandan R., Srinivasan P., Dinesh D., Babu G., Sellamuthu S.,
Volume : 2   Issue : 1,   Year : 2010           Downloads : 1083

IDENTIFICATION OF T-CELL EPITOPE FOR PROTECTIVE ANTIGEN AND LETHAL FACTOR OF Bacillus anthracis - AN IMMUNOINFORMATICS APPROACH
ANURAJ NAYARISSERI, MUKESH YADAV, SHEAZA AHMED, JYOTI SAHU, PRIYANKA GUPTA, RACHNA CHOURASIA, DEEPTI MITTAL,
Volume : 4   Issue : 1,   Year : 2012           Downloads : 1076

Protein networks in diseases
Kayarkar N. A., Durgude S. G., Maurya B.D., Pawar S. V., Chate P. B.,
Volume : 1   Issue : 2,   Year : 2009           Downloads : 1060

SYNTHESIS, STRUCTURAL, AND BIOLOGICAL SCREENING OF SOME NEW ORGANOBISMUTH COMPOUNDS
TEWARI I.C., TIWARI V.K., SUSHMA RANI,
Volume : 3   Issue : 2,   Year : 2011           Downloads : 1059

MOLECULAR CHARACTERIZATION OF EXTENDED-SPECTRUM Î’- LACTAMASES PRODUCING CTX-M-15 FROM GRAM NEGATIVE BACTERIA ISOLATED FROM PEDIATRIC AND NEONATAL INTENSIVE CARE UNIT
JADHAV S.V., JADHAV R., GANDHAM N., MISRA R., SINGH P., UJAGARE M., ANGADI K., VYAWAHARE C.,
Volume : 4   Issue : 2,   Year : 2012           Downloads : 1059

PHARMACOGENOINFORMATICS: MODELING OF P-GLYCOPROTEIN AND NOVEL APPROACH OF In Silico DRUG DESIGNING BASED ON GENETIC VARIATION OF MDR1 GENE INVOLVED IN STATIN RESISTANCE
ANJANA MUNSHI, SAI BABU M., VENKATESWARA RAO A., LAKSHMAN TEJA G., SUBASH KAUL, JYOTHY A.,
Volume : 4   Issue : 1,   Year : 2012           Downloads : 1051

Analog based pharmacophore strategy to identify novel leukotriene a4 hydrolase (LTA4H) inhibitors
Kranthi Raj K., Pathak L.P., Muttineni Ravikumar, Ramachandrana D.,
Volume : 2   Issue : 2,   Year : 2010           Downloads : 1047

Prediction of antigenic peptides of LTx5 toxin from Lasiodora sp. IBSP8539
Gomase V.S., Shankar S., Gangawane A.K., Sherkhane A.S.,
Volume : 1   Issue : 1,   Year : 2009           Downloads : 1046

Human proteome: New research technologies for cancer research
More M.K., Nair V.K., Thikekar V.P., Sawant J.J., Ravidhone Y., Patil A., Paul Andrea.,
Volume : 1   Issue : 2,   Year : 2009           Downloads : 1044

Active site binding interactions of β-carboline derivative for HIV reverse transcriptase, protease and integrase
Prabha Garg, Rajender Kumar,
Volume : 2   Issue : 2,   Year : 2010           Downloads : 1042

THE CHOICE OF PHASE I BAYESIAN ADAPTIVE DESIGNS IN CHINA
PAN H., JI Y., CHEN Z., LI C., XIA J.,
Volume : 5   Issue : 1,   Year : 2013           Downloads : 1038

In vitro studies on anti asthmatic, analgesic and anti convulsant activities of the medicinal plant Bryonia laciniosa.Linn
Vijay D., Jayarama Reddy, Gnanasekaran D., Ranganathan T.V.,
Volume : 2   Issue : 2,   Year : 2010           Downloads : 1034

Protein Based Drug Discovery
Joshi B., Gupta G., Gupta N., Gupta M., Trivedi S., Patil P., Jhadav A., Vamsi K.K., Khairnar Y., Boraste A., Mujapara A.,
Volume : 1   Issue : 2,   Year : 2009           Downloads : 1028

AN INVESTIGATION ON CYTOTOXIC AND ANTIOXIDANT PROPERTIES OF CLITORIA TERNATEA L.
VIDHYA RAMASWAMY, NEETHU VARGHESE, ANCY SIMON,
Volume : 3   Issue : 1,   Year : 2011           Downloads : 1028

A LINEAR QSAR AND DOCKING APPROACH TO MODEL INHIBITORY ACTIVITY OF 2-ARYLBENZOXAZOLE DERIVATIVES AS CHOLESTERYL ESTER TRANSFER PROTEIN (CETP) INHIBITORS
MUKESH YADAV, ANURAJ NAYARISSERI, SHOBHA JOSHI, ANKITA GUPTA, PURVA HOLKAR, ASHISH RAJPUT,
Volume : 3   Issue : 1,   Year : 2011           Downloads : 1026

IN-SILICO ANALYSIS OF QUINOXALINE LIGAND CONFORMATIONS ON 2BB9: HIV-1 PROTEASE
ARUNKUMAR V.A., KESHAV MOHAN,
Volume : 4   Issue : 2,   Year : 2012           Downloads : 1004

INVIVO EVALUATION OF THE EFFECTS OF Allium sativum ON THE PHARMACOKINETIC PARAMETERS OF CIPROFLOXACIN AND ISONIAZID.
NDUKA S.O., OKONTA J.M., ESIMONE C.O.,
Volume : 4   Issue : 1,   Year : 2012           Downloads : 994

Proteomics based prediction of antigenicity of iberiotoxin from eastern Indian scorpion
Gomase V.S., Phadnis A.C., Waghmare Somnath,
Volume : 1   Issue : 1,   Year : 2009           Downloads : 978

HISTOLOGICAL STUDY ON THE EFFECT OF Arabidopsis thaliana EXTRACT ON ALLOXAN-INDUCED DIABETIC INFERTILITY MICE
TAHA M.A., AHMED S.J., RASHID K.I.,
Volume : 6   Issue : 1,   Year : 2014           Downloads : 976

THE CHALLENGES OF OPHTHALMIC DRUG DELIVERY: A REVIEW
HEMING T., SINGH V., AHMAD R.,
Volume : 3   Issue : 1,   Year : 2011           Downloads : 974

OPTIMIZED COMBINATIONS OF OCIMUM ESSENTIAL OILS INHIBIT GROWTH OF FOUR Candida albicans
HZOUNDA F.J.B., JAZET D.P.M., BAKARNGA V.I., NGO MBACK M.N.L., ZEUKO'O M.E., FALL A.D., BASSENE E., FEKAM B.F.,
Volume : 6   Issue : 1,   Year : 2014           Downloads : 968

Particulate vaccine for bacterial diseases
Hariprasad O., Gopinath V.P., Navya A., Yugandhar V.G., Sarma P.V.G.K,
Volume : 2   Issue : 2,   Year : 2010           Downloads : 948

BIOCHEMICAL CHARACTERIZATION OF VOLATILE SECONDARY METABOLITES PRODUCED BY Burkholderia gladioli pv. agaricicola
ELSHAFIE H.S., BUFO S.A., RACIOPPI R., CAMELE I.,
Volume : 5   Issue : 1,   Year : 2013           Downloads : 943

ANTITUMOR ACTIVITY OF BIOMOLECULES: A BRIEF REVIEW
SOUZA P.O., RITTER M., BRAGANHOL E., PEREIRA C.M.P.,
Volume : 6   Issue : 1,   Year : 2014           Downloads : 942

Immunoproteomics approach for prediction of antigenic epitope of Tertiapin from Apis mellifera
Gomase V. S., Phadnis A. C., Ghatak A.A.,
Volume : 1   Issue : 1,   Year : 2009           Downloads : 931

THE COMPUTER AIDED DRUG DESIGNING FOR THE DIABETIC TARGET: ALDOSE REDUCTASE
DALAL H.,
Volume : 6   Issue : 1,   Year : 2014           Downloads : 912

INTRODUCING "SYNTHESIS ROUTE-BASED HIT IDENTIFICATION APPROACH" AS A TOOL IN MEDICINAL CHEMISTRY AND ITS APPLICATION IN INVESTIGATING THE ANTIPROLIFERATIVE AND ANTIMICROBIAL EFFECTS OF 2- AMINOPYRIMIDINE DERIVATIVES
FARZAD KOBARFARD, SHOHREH MOHEBBI, FARSHAD H. SHIRAZI, SEYED HESAMEDIN SHARIFNIA,
Volume : 3   Issue : 2,   Year : 2011           Downloads : 895

IN SILICO DESIGN OF Butea monosperma FLORAL DERIVED COMPOUNDS AND ITS INHIBITORY EFFECT ON β-CATENIN, GSK-3β AND APC COMPLEX PROTEINS IN COLORECTAL CANCER
NAVANEETHAKRISHNAN P., PRASHANTHA C.N., BOOPATHI S., SABITHA R., MATHAN G.,
Volume : 5   Issue : 1,   Year : 2013           Downloads : 866

RELATIONSHIP BETWEEN QUINOLONE STRUCTURE AND MINIMAL INHIBITORY CONCENTRATION OF BACTERIAL STRAINS
M. MARCZAK, T. GRABOWSKI,
Volume : 7   Issue : 1,   Year : 2015           Downloads : 705

WOUND HEALING: CURRENT UNDERSTANDING AND FUTURE PROSPECT
AJAY KUMAR SHARMA, VIGHNESH SUNDER, M.H. YASHAVARDDHAN, SANDEEP KUMAR SHUKLA,
Volume : 8   Issue : 1,   Year : 2017           Downloads : 506

MOLECULAR DOCKING OF ALKALOID COMPOUND SA2014 FROM MARINE SPONGES Cinachyrella anomala TOWARDS P53 PROTEIN
AWIK PUJI DYAH NURHAYATI, MARDI SANTOSO, EDWIN SETIAWAN, FITRI LIANINGSIH,
Volume : 8   Issue : 1,   Year : 2017           Downloads : 503